Bilaid A1

Bilaid A1

$280.00 - 1 mg

$980.00 - 5 mg

All prices in Australian dollars

Code
BIA-B2275
CAS #
2393866-02-7
Molecular Formula
C28H39N5O4
Molecular Weight
509.7
Purity
>95% by HPLC
Long Term Storage
-20°C
Solubility
Soluble in methanol or DMSO

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Application Notes

Bilaid A1 (FvVf-NH2) is the semi-synthetic analogue of Bilaid A, an unusual tetrapeptide isolated from an Australian estuarine isolate of Penicillium sp. MST-MF667. Conversion of the terminal carboxylate to its corresponding amide enhanced the μ-​opioid agonist potency leading to the design of more potent analogues, bilorphin and bilactorphin.

References

  • A tetrapeptide class of biased analgesics from an Australian fungus targets the μ-​opioid receptor. Dekan Z. et al. Proc Nat Acad Sci. 2019, 116, 22535.

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